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環(huán)多肽試劑:cyclo(RGDFK(DOTA)),整合素 αvβ3 抑制劑

2023-06-19 15:18 作者:新研之家  | 我要投稿

PART1----試劑基礎(chǔ)信息:

cyclo(RGDFK(DOTA)),環(huán)多肽試劑
Product structure:

Product specifications:
1.CAS No:N/A
2.Molecular formula:N/A
3.Molecular weight:N/A
4.Packaging specification:1g、5g、10g, flexible packaging, including 100mg packaging and 500mg 1g and 5g large packaging
5.Appearance color:The product is a solid or viscous liquid, depending on the molecular weight of PEG
6.Dissolution conditions:Soluble in most organic solvents, such as DCM, DMF, DMSO, THF, etc., with good solubility in water

7.Stability:-1 year at 20 ° C, dry and dark.

8.Supplier:陜西新研博美生物科技有限公司

PART2----試劑反應(yīng)特點(diǎn):

cyclo(RGDFK(DOTA))屬于環(huán)多肽試劑,Cyclo(-RGDfK) 是有效,選擇性的整合素 αvβ3 抑制劑,其 IC50 值為 0.94 nM。不同標(biāo)記物可以對肽進(jìn)行修飾,例如烷基化太、PEG修飾肽、雙標(biāo)記修飾肽、馬來酰亞胺基修飾肽、二硫鍵環(huán)肽、酰胺鍵環(huán)肽等一系列的。

PART3----同類型試劑整理:

CAS:782423-00-1?,英文名:Gd-DO3A-Butylamine
CAS:72573-82-1,英文名:Gd-DOTA
CAS:2126179-26-6,英文名:Gd-p-SCN-Bn-DOTA
CAS:1349103-97-4,英文名:Ho-Maleimido-DOTA
CAS:2126179-28-8,英文名:Ho-p-SCN-Bn-DOTA
CAS:78063-83-9,英文名:Tm-DOTA
CAS:2126179-30-2,英文名:Tm-DOTMA
CAS:30859-88-8,英文名:Tm-DOTP
CAS:1552305-24-4,英文名:Tm-Maleimido-DOTA
CAS:2126179-32-4,英文名:Tm-p-SCN-Bn-DOTA
CAS:162148-45-0,英文名:Bis-CBZ-Cyclen
CAS:162148-48-3,英文名:DO2A-tert-butyl ester
CAS:122555-91-3,英文名:DO3A-tert-butyl ester , DO3A-tBu-ester
CAS:174137-97-4,英文名:NO2A-(t-Bu ester)
CAS:175854-39-4,英文名:Tris-BOC-Cyclen
CAS:1006711-09-5,英文名:Maleimide-DOTA

PART4----使用保存說明:

1.Matters for use:

It is sensitive to light and temperature. In order to use the reagent effectively, the material should always be kept in a low temperature dry condition, away from light, and avoid frequent thawing and freezing.
2.storage conditions:
Store at - 20 ℃ as much as possible. If conditions permit, the material can be treated under inert gas to obtain better stability of the reagent.

以上陜西新研博美生物科技有限公司MISS.wu編輯的試劑信息僅用于科學(xué)研究或者工業(yè)應(yīng)用等非醫(yī)療目的,非藥用,非食用。接受各種復(fù)雜定制服務(wù),合成的Monodispersed PEGs除了有更多樣的基團(tuán)還可以提供各種不同數(shù)量的PEG的產(chǎn)品。

環(huán)多肽試劑:cyclo(RGDFK(DOTA)),整合素 αvβ3 抑制劑的評論 (共 條)

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